Orfadin

Product NDC
66658-105
11-digit product format
666580105
Labeler code
66658
Product ID
66658-105_f9c6cef5-fb71-4cb0-9793-5c23ac04572e
Type
HUMAN PRESCRIPTION DRUG
Nonproprietary name
Nitisinone
Dosage form
CAPSULE
Route
ORAL
Labeler
SWEDISH ORPHAN BIOVITRUM AB (PUBL)
Application
NDA021232
Marketing category
NDA
Marketing start
2016-07-01
Substance
NITISINONE
Active strength
5 mg/1
Pharmacologic classes
4-Hydroxyphenyl-Pyruvate Dioxygenase Inhibitor [EPC], Cytochrome P450 2C9 Inhibitors [MoA], Cytochrome P450 2E1 Inducers [MoA], Hydroxyphenylpyruvate Dioxygenase Inhibitors [MoA], Organic Anion Transporter 1 Inhibitors [MoA], Organic Anion Transporter 3 Inhibitors [MoA]
NDC exclude flag
No
Listing certified through
2026-12-31
Current FDA listing
Yes

Source provenance: Browse the complete Orange Book source catalog · source snapshot 42.

Orange Book products#

Current product rows page 1 of 1 · 4 matching rows.

Application-product, Trade name, Ingredient table
Application-productTrade nameIngredientStrengthDosage form / routeTE codesRLD / RSApproval date
N021232-001ORFADINNITISINONE2MGCAPSULE / ORALABRLD2002-01-18
N021232-002ORFADINNITISINONE5MGCAPSULE / ORALABRLD2002-01-18
N021232-003ORFADINNITISINONE10MGCAPSULE / ORALABRLD2002-01-18
N021232-004ORFADINNITISINONE20MGCAPSULE / ORALABRLD, RS2016-06-13

Therapeutic equivalence codes#

Current TE-code rows page 1 of 1 · 4 matching rows.

Application-product, TE code table
Application-productTE code
N021232-001AB
N021232-002AB
N021232-003AB
N021232-004AB

Observed Orange Book product history#

Observed FDA ZIP history: Each table is queried independently by exact application/product key from successfully parsed Orange Book snapshots. Capture times identify archived source observations; absence or a change between snapshots is not inferred. FDA publication files that were not recoverable as structured ZIP data are not represented as states.

Product history page 1 of 5 · 168 observed states.

Captured, Edition, Application-product table
CapturedEditionApplication-productTrade nameStrengthDosage form / routeProduct TE source textRLD / RSApproval dateSource SHA-256
2026-08-18 06:07:402026-07N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-18caaa826d4ba7…
2026-08-18 06:07:402026-07N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-18caaa826d4ba7…
2026-08-18 06:07:402026-07N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-18caaa826d4ba7…
2026-08-18 06:07:402026-07N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-13caaa826d4ba7…
2026-02-19 14:30 UTC2026-02N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-18011fe1cb6892…
2026-02-19 14:30 UTC2026-02N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-18011fe1cb6892…
2026-02-19 14:30 UTC2026-02N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-18011fe1cb6892…
2026-02-19 14:30 UTC2026-02N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-13011fe1cb6892…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-1831067a03dcf5…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-1831067a03dcf5…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-1831067a03dcf5…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-1331067a03dcf5…
2025-08-23 18:47 UTC2025-08N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-186a471c1ec25d…
2025-08-23 18:47 UTC2025-08N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-186a471c1ec25d…
2025-08-23 18:47 UTC2025-08N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-186a471c1ec25d…
2025-08-23 18:47 UTC2025-08N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-136a471c1ec25d…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-18fd3edfee7708…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-18fd3edfee7708…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-18fd3edfee7708…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-13fd3edfee7708…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-18b8a1b40f171c…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-18b8a1b40f171c…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-18b8a1b40f171c…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-13b8a1b40f171c…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-1803ed91905a0d…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-1803ed91905a0d…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-1803ed91905a0d…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-1303ed91905a0d…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-182680178bc6a6…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-182680178bc6a6…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-182680178bc6a6…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-132680178bc6a6…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-185bbf6a4d5a75…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-185bbf6a4d5a75…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-185bbf6a4d5a75…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-135bbf6a4d5a75…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-001ORFADIN2MGCAPSULE / ORALABRLD2002-01-18d8e5a09893c0…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-002ORFADIN5MGCAPSULE / ORALABRLD2002-01-18d8e5a09893c0…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-003ORFADIN10MGCAPSULE / ORALABRLD2002-01-18d8e5a09893c0…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-004ORFADIN20MGCAPSULE / ORALABRLD, RS2016-06-13d8e5a09893c0…

Observed Orange Book normalized TE history#

Normalized TE history page 1 of 4 · 148 observed states.

Captured, Edition, Application-product table
CapturedEditionApplication-productTE codeOrderSource SHA-256
2026-08-18 06:07:402026-07N021232-001AB1caaa826d4ba7…
2026-08-18 06:07:402026-07N021232-002AB1caaa826d4ba7…
2026-08-18 06:07:402026-07N021232-003AB1caaa826d4ba7…
2026-08-18 06:07:402026-07N021232-004AB1caaa826d4ba7…
2026-02-19 14:30 UTC2026-02N021232-001AB1011fe1cb6892…
2026-02-19 14:30 UTC2026-02N021232-002AB1011fe1cb6892…
2026-02-19 14:30 UTC2026-02N021232-003AB1011fe1cb6892…
2026-02-19 14:30 UTC2026-02N021232-004AB1011fe1cb6892…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-001AB131067a03dcf5…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-002AB131067a03dcf5…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-003AB131067a03dcf5…
2025-12-14 10:44 UTC · 2 captures of this ZIP2025-12N021232-004AB131067a03dcf5…
2025-08-23 18:47 UTC2025-08N021232-001AB16a471c1ec25d…
2025-08-23 18:47 UTC2025-08N021232-002AB16a471c1ec25d…
2025-08-23 18:47 UTC2025-08N021232-003AB16a471c1ec25d…
2025-08-23 18:47 UTC2025-08N021232-004AB16a471c1ec25d…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-001AB1fd3edfee7708…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-002AB1fd3edfee7708…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-003AB1fd3edfee7708…
2025-03-22 03:13 UTC · 3 captures of this ZIP2025-03N021232-004AB1fd3edfee7708…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-001AB1b8a1b40f171c…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-002AB1b8a1b40f171c…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-003AB1b8a1b40f171c…
2025-02-26 10:13 UTC · 3 captures of this ZIP2025-02N021232-004AB1b8a1b40f171c…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-001AB103ed91905a0d…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-002AB103ed91905a0d…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-003AB103ed91905a0d…
2025-01-19 17:59 UTC · 7 captures of this ZIP2025-01N021232-004AB103ed91905a0d…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-001AB12680178bc6a6…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-002AB12680178bc6a6…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-003AB12680178bc6a6…
2024-12-13 21:23 UTC · 2 captures of this ZIP2024-12N021232-004AB12680178bc6a6…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-001AB15bbf6a4d5a75…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-002AB15bbf6a4d5a75…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-003AB15bbf6a4d5a75…
2024-09-14 05:58 UTC · 2 captures of this ZIP2024-09N021232-004AB15bbf6a4d5a75…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-001AB1d8e5a09893c0…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-002AB1d8e5a09893c0…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-003AB1d8e5a09893c0…
2024-11-08 22:44 UTC · 3 captures of this ZIP2024-11N021232-004AB1d8e5a09893c0…

Observed Orange Book exclusivity history#

Captured, Edition, Application-product table
CapturedEditionApplication-productExclusivity codeExpirationSource SHA-256
2019-12-13 00:20 UTC2019-12N021232-001D-1692020-09-0174a2ff9319b5…
2019-12-13 00:20 UTC2019-12N021232-002D-1692020-09-0174a2ff9319b5…
2019-12-13 00:20 UTC2019-12N021232-003D-1692020-09-0174a2ff9319b5…
2019-12-13 00:20 UTC2019-12N021232-004D-1692020-09-0174a2ff9319b5…
2020-12-22 03:56 UTC2020-12N021232-001D-1692020-09-018869cabd3fbd…
2020-12-22 03:56 UTC2020-12N021232-002D-1692020-09-018869cabd3fbd…
2020-12-22 03:56 UTC2020-12N021232-003D-1692020-09-018869cabd3fbd…
2020-12-22 03:56 UTC2020-12N021232-004D-1692020-09-018869cabd3fbd…
2020-11-12 02:37 UTC2020-11N021232-001D-1692020-09-01c0c555d07b60…
2020-11-12 02:37 UTC2020-11N021232-002D-1692020-09-01c0c555d07b60…
2020-11-12 02:37 UTC2020-11N021232-003D-1692020-09-01c0c555d07b60…
2020-11-12 02:37 UTC2020-11N021232-004D-1692020-09-01c0c555d07b60…
2019-12-14 00:12 UTC2019-12N021232-001D-1692020-09-013f01610625f2…
2019-12-14 00:12 UTC2019-12N021232-002D-1692020-09-013f01610625f2…
2019-12-14 00:12 UTC2019-12N021232-003D-1692020-09-013f01610625f2…
2019-12-14 00:12 UTC2019-12N021232-004D-1692020-09-013f01610625f2…
2019-09-15 20:21 UTC2019-09N021232-001D-1692020-09-01b00525d2431f…
2019-09-15 20:21 UTC2019-09N021232-002D-1692020-09-01b00525d2431f…
2019-09-15 20:21 UTC2019-09N021232-003D-1692020-09-01b00525d2431f…
2019-09-15 20:21 UTC2019-09N021232-004D-1692020-09-01b00525d2431f…
2019-07-19 19:46 UTC2019-07N021232-001D-1692020-09-01ea99ee380514…
2019-07-19 19:46 UTC2019-07N021232-002D-1692020-09-01ea99ee380514…
2019-07-19 19:46 UTC2019-07N021232-003D-1692020-09-01ea99ee380514…
2019-07-19 19:46 UTC2019-07N021232-004D-1692020-09-01ea99ee380514…

Additional Listing Data#

Finished product
Yes
Brand name base
Orfadin
Listing expiration
2026-12-31

Active Ingredients#

Ingredient, Strength table
IngredientStrength
NITISINONE5 mg/1

Harmonized UNII identifiers#

UNII identifiers page 1 of 1 · 1 matching rows.

Identifier, FDA.report destination table
IdentifierFDA.report destination
K5BN214699Internal UNII lookup

Harmonized RxCUI identifiers#

RxCUI identifiers page 1 of 1 · 8 matching rows.

Identifier, FDA.report destination table
IdentifierFDA.report destination
351173Internal RxNorm lookup
351174Internal RxNorm lookup
351175Internal RxNorm lookup
352119Internal RxNorm lookup
352120Internal RxNorm lookup
352121Internal RxNorm lookup
1798999Internal RxNorm lookup
1799001Internal RxNorm lookup

Harmonized SPL set identifiers#

SPL set identifiers page 1 of 1 · 1 matching rows.

Identifier, FDA.report destination table
IdentifierFDA.report destination
5d449b73-d503-4132-b978-d890491975dfAvailable on FDA.report

DailyMed Product Concepts#

Product concept, Relation, Version table
Product conceptRelationVersionEffective
30289e20-d00d-4455-8aae-af8add8f10eeProduct name420240529
5b3e65b0-2e25-4346-b6a5-74172e0cd130Product name120170824
689eee6a-c9bd-41ef-86ac-b494143eb282Product name220160804

DailyMed Package Descriptions#

Package NDC, Product, Description table
Package NDCProductDescriptionFormQuantityStrengthSPL version
66658-105-60Orfadin1 in 1 CARTONCAPSULE114
66658-105-60Orfadin60 in 1 BOTTLE, PLASTICCAPSULE6014

DailyMed Billing Units#

Package NDC, Billing unit, Product NDC table
Package NDCBilling unitProduct NDCDailyMed indexing SPLSPL versionEffective
66658-105-60EA - Each66658-105612db024-cb21-4ec9-8dde-e7bcf4b1052812014-04-03

DailyMed Socrata Ingredients#

DailyMed Dashboard NDC Coverage#

NDC, Dashboard title, SPL version table
NDCDashboard titleSPL versionValidationDashboard ZIP
66658-105ORFADIN (NITISINONE) CAPSULE [SWEDISH ORPHAN BIOVITRUM AB (PUBL)]14Current NDC, Legacy NDC, 2 package rows20220612_5d449b73-d503-4132-b978-d890491975df.zip

openFDA label cross-check#

OpenFDA label data provides additional search and identifier links. DailyMed’s Structured Product Label is the canonical label on FDA.report. Matching records are deduplicated before they are shown below.

Matched openFDA labels page 1 of 1 · 1 matching rows.

Brand, Generic, Manufacturer table
BrandGenericManufacturerSPL set IDEffective dateAvailable safety fieldsJoin
OrfadinNITISINONESWEDISH ORPHAN BIOVITRUM AB (PUBL)5d449b73-d503-4132-b978-d890491975df2021-11-30Warnings, Adverse reactionsExact identifier
application applno (NDA): 021232
application number: NDA021232
ndc (product): 66658-105

DailyMed RxNorm Mappings#

RxCUI, RxNorm string, TTY table
RxCUIRxNorm stringTTYDailyMedSPL version
351175nitisinone 10 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
351173nitisinone 2 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
1798999nitisinone 20 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
351174nitisinone 5 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
352121Orfadin 10 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
352119Orfadin 2 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
1799001Orfadin 20 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
352120Orfadin 5 MG Oral CapsulePSN5d449b73-d503-4132-b978-d890491975df14
352121nitisinone 10 MG Oral Capsule [Orfadin]SBD5d449b73-d503-4132-b978-d890491975df14
352119nitisinone 2 MG Oral Capsule [Orfadin]SBD5d449b73-d503-4132-b978-d890491975df14
1799001nitisinone 20 MG Oral Capsule [Orfadin]SBD5d449b73-d503-4132-b978-d890491975df14
352120nitisinone 5 MG Oral Capsule [Orfadin]SBD5d449b73-d503-4132-b978-d890491975df14
351175nitisinone 10 MG Oral CapsuleSCD5d449b73-d503-4132-b978-d890491975df14
351173nitisinone 2 MG Oral CapsuleSCD5d449b73-d503-4132-b978-d890491975df14
1798999nitisinone 20 MG Oral CapsuleSCD5d449b73-d503-4132-b978-d890491975df14
351174nitisinone 5 MG Oral CapsuleSCD5d449b73-d503-4132-b978-d890491975df14
352121Orfadin 10 MG Oral CapsuleSY5d449b73-d503-4132-b978-d890491975df14
352119Orfadin 2 MG Oral CapsuleSY5d449b73-d503-4132-b978-d890491975df14
1799001Orfadin 20 MG Oral CapsuleSY5d449b73-d503-4132-b978-d890491975df14
352120Orfadin 5 MG Oral CapsuleSY5d449b73-d503-4132-b978-d890491975df14

Packages#

Package NDC, 11-digit format, Description table
Package NDC11-digit formatDescriptionMarketing startMarketing endSampleExclude flagStatus
66658-105-60666580105601 BOTTLE, PLASTIC in 1 CARTON (66658-105-60) / 60 CAPSULE in 1 BOTTLE, PLASTIC2016-07-010000-00-00NoNoCurrent